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dc.contributor.authorTu, Songzh_CN
dc.contributor.authorXie, Ya-Qiangzh_CN
dc.contributor.authorGui, Si-Zhezh_CN
dc.contributor.authorYe, Li-Yizh_CN
dc.contributor.authorHuang, Zi-Longzh_CN
dc.contributor.authorHuang, Yi-Bingzh_CN
dc.contributor.authorChe, Li-Mingzh_CN
dc.contributor.author叶李艺zh_CN
dc.date.accessioned2015-07-22T03:21:15Z
dc.date.available2015-07-22T03:21:15Z
dc.date.issued2014-05-01zh_CN
dc.identifier.citationBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014,24(9):2173-2176zh_CN
dc.identifier.otherWOS:000334337100029zh_CN
dc.identifier.urihttps://dspace.xmu.edu.cn/handle/2288/89313
dc.descriptionNational Nature Science Foundation of China [21106119]; Fundamental Research Funds for the Central Universities, PR China [2011121019]zh_CN
dc.description.abstractTwenty-one novel benzothiophene-substituted oxime ether strobilurins, which employed a benzothiophene group to stabilise the E-styryl group in Enoxastrobin (an unsaturated oxime strobilurin fungicide developed by Shenyang Research Institute of Chemical Industry, China) were designed and synthesised. The biological assay indicated that most compounds exhibited good or excellent fungicidal activities, especially against Colletotrichum lagenarium and Puccinia sorghi Schw. In addition, methyl 3-methoxy-propenoate oxime ethers and N-methoxy-carbamic acid methyl esters exhibited good in vivo fungicidal activities against Erysiphe graminis, Colletotrichum lagenarium and Puccinia sorghi Schw. under the tested concentrations. Notably, (E, E)-methyl 3-methoxy-2-(2-((((6-chloro-1-(1H-benzo[b] thien-2-yl)ethylidene)amino)oxy) methyl) phenyl) propenoate (5E) exhibited more potent in vivo fungicidal activities against nearly all of the tested fungi at a concentration of 0.39 mg/L compared to Enoxastrobin. (C) 2014 Elsevier Ltd. All rights reserved.zh_CN
dc.language.isoen_USzh_CN
dc.publisherPERGAMON-ELSEVIER SCIENCE LTDzh_CN
dc.source.urihttp://dx.doi.org/10.1016/j.bmcl.2014.03.024zh_CN
dc.subjectBIOLOGICAL-ACTIVITIESzh_CN
dc.subjectNATURAL-PRODUCTSzh_CN
dc.subjectCROP PROTECTIONzh_CN
dc.subjectLOCKED ANALOGSzh_CN
dc.subjectCHEMISTRYzh_CN
dc.subjectDESIGNzh_CN
dc.subjectAGENTSzh_CN
dc.titleSynthesis and fungicidal activities of novel benzothiophene-substituted oxime ether strobilurinszh_CN
dc.typeArticlezh_CN


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